SCHEMBL2827012

SCHEMBL2827012

Cc1nccc(NC(=O)Oc2nc(C)sc2Nc2cccc(C(N)=O)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.47
LCK P06239 1/20 0.44
FYN P06241 1/20 0.44
YES1 P07947 1/20 0.44
LYN P07948 1/20 0.44
FGR P09769 1/20 0.44
EPHA1 P21709 1/20 0.44
EPHA2 P29317 1/20 0.44
EPHA3 P29320 1/20 0.44
EPHB2 P29323 1/20 0.44
CSK P41240 1/20 0.44
TXK P42681 1/20 0.44
SYK P43405 1/20 0.44
BLK P51451 1/20 0.44
BMX P51813 1/20 0.44
EPHB3 P54753 1/20 0.44
EPHA5 P54756 1/20 0.44
EPHA4 P54764 1/20 0.44
BTK Q06187 1/20 0.44
TYRO3 Q06418 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2831282 0.87 NPC1 (0.43)
SCHEMBL2826236 0.86 GRM5 (0.49) ROCK1LCKFYNYES1LYN
SCHEMBL2826867 0.84 CDK4 (0.45)
SCHEMBL2830181 0.84 ROCK1 (0.46) ROCK1LCKSYKTYRO3
SCHEMBL2833176 0.84 SORT1 (0.41)
SCHEMBL2826585 0.83 GRM5 (0.52)
SCHEMBL2830050 0.83 BRAF (0.46)
SCHEMBL2830257 0.81 GRM5 (0.50)
SCHEMBL2829325 0.78 JAK2 (0.41)
SCHEMBL2828980 0.78 SORT1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed