SCHEMBL28276502

SCHEMBL28276502

COC(=O)c1ccc(Oc2ccccc2F)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.67
KMT2A Q03164 2/20 0.61
ALDH1A1 P00352 1/20 0.61
LPAR1 Q92633 8/20 0.53
LPAR5 Q9H1C0 8/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
TSHR P16473 1/20 0.52
MAPT P10636 5/20 0.51
RAB9A P51151 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 3/20 0.51
HTT P42858 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
KDM4E B2RXH2 1/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
LMNA P02545 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11411879 0.88 CA1 (0.62) KMT2AALDH1A1LPAR1LPAR5CA1
SCHEMBL9242685 0.85 RAB9A (0.65) PARP10KMT2AALDH1A1LPAR1LPAR5
SCHEMBL15669422 0.84 NPC1 (0.53) PARP10KMT2AALDH1A1CA1CA2
SCHEMBL16507371 0.84 LPAR1 (0.79) LPAR1LPAR5
SCHEMBL9762806 0.83 PARP10 (0.71) PARP10LPAR1LPAR5MAPTRAB9A
SCHEMBL16506947 0.83 LPAR1 (0.82) LPAR1LPAR5
SCHEMBL10437240 0.83 PARP10 (0.65) PARP10KMT2AALDH1A1LPAR1LPAR5
SCHEMBL8782253 0.82 SLC6A3 (0.61) KMT2AALDH1A1LPAR1LPAR5CA1
SCHEMBL1191950 0.82 TDP1 (0.68) KMT2AALDH1A1LPAR1LPAR5CA1
SCHEMBL24209453 0.82 PARP10 (0.60) PARP10LPAR1LPAR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641897-A Bcl-2 selective depressant and its preparation and use 北京赛林泰医药技术有限公司 2019-04-16 CN disclosed
CN-109311860-A For treating or preventing the Xanthone derivative of hepatitis type B virus disease 豪夫迈·罗氏有限公司 2019-02-05 CN disclosed