SCHEMBL28280295

SCHEMBL28280295

NC(=O)c1cccc(NC([O])=O)c1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
PARP1 P09874 16/20 0.61
PARP10 Q53GL7 12/20 0.61
PARP15 Q460N3 7/20 0.61
PARP14 Q460N5 4/20 0.61
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850002 0.86 MEN1 (0.67) MEN1KMT2APARP1PARP10PARP15
SCHEMBL4893340 0.85 PARP1 (0.66) MEN1KMT2APARP1PARP10PARP15
SCHEMBL5425792 0.85 MEN1 (0.65) MEN1KMT2APARP1PARP10PARP15
SCHEMBL895009 0.83 PARP1 (0.63) MEN1KMT2APARP1PARP10PARP15
SCHEMBL408480 0.83 PARP1 (0.63) MEN1KMT2APARP1PARP10PARP15
SCHEMBL4531507 0.83 ALDH1A1 (0.71) MEN1KMT2APARP1PARP10PARP15
SCHEMBL895690 0.83 MEN1 (0.63) MEN1KMT2APARP1PARP10PARP15
SCHEMBL29761319 0.83 PARP1 (0.63) MEN1KMT2APARP1PARP10PARP15
SCHEMBL9921486 0.82 MEN1 (0.61) MEN1KMT2APARP1PARP10PARP15
SCHEMBL18671651 0.81 KMT2A (0.87) MEN1KMT2APARP1PARP10PARP15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108138177-B The combination of Dbait molecule and PARP inhibitor is used for the purposes for the treatment of cancer 法国居里学院 2019-03-19 CN disclosed