SCHEMBL2828409

SCHEMBL2828409

CCOC(=O)c1cc(Br)cc(OCCCCCBr)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 1/20 0.47
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
ESR1 P03372 4/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
BRD4 O60885 1/20 0.41
BRD2 P25440 1/20 0.41
CREBBP Q92793 1/20 0.41
AKR1C4 P17516 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41
SMPD1 P17405 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826323 0.87 ALDH1A1 (0.53) PLA2G2AESR1TDP1
SCHEMBL22868140 0.85 L3MBTL1 (0.48) PLA2G2ACA12CA1CA2CA7
SCHEMBL2826636 0.85 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL288382 0.85 BRD4 (0.53) CA12CA1CA2CA7CA9
SCHEMBL2822392 0.84 CA12 (0.46) PLA2G2ACA12CA1CA2CA7
SCHEMBL4727671 0.83 PLA2G2A (0.54) PLA2G2ACA12CA1CA2CA7
SCHEMBL20958112 0.82 PLA2G2A (0.69) PLA2G2ACA12CA1CA2CA7
SCHEMBL5491044 0.82 PLA2G2A (0.64) PLA2G2ACA12CA1CA2CA7
SCHEMBL9387912 0.82 PLA2G2A (0.69) PLA2G2ACA12CA1CA2CA7
SCHEMBL2821784 0.82 ALDH1A1 (0.52) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069504-A1 (3-OXO)PYRIDIN-4-YLUREA DERIVATIVES AS PDE4 INHIBITORS ALMIRALL, S.A. (ES) 2010-06-24 WO disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed