SCHEMBL28291583

SCHEMBL28291583

O=C(O)c1ccc2c(c1)CCCN2C[SH](=O)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
HDAC1 Q13547 8/20 0.47
HDAC6 Q9UBN7 8/20 0.47
HDAC8 Q9BY41 6/20 0.47
HDAC3 O15379 2/20 0.47
HDAC4 P56524 2/20 0.47
HDAC7 Q8WUI4 2/20 0.47
HDAC2 Q92769 2/20 0.47
HDAC11 Q96DB2 2/20 0.47
HDAC9 Q9UKV0 2/20 0.47
HDAC5 Q9UQL6 2/20 0.47
CYP2C19 P33261 1/20 0.47
PDK1 Q15118 1/20 0.47
PDK2 Q15119 1/20 0.47
PDK3 Q15120 1/20 0.47
PDK4 Q16654 1/20 0.47
MCL1 Q07820 2/20 0.46
HDAC10 Q969S8 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
KDM4E B2RXH2 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20178649 0.82 ALDH1A1 (0.52) ALDH1A1HDAC1HDAC6HDAC8HDAC3
SCHEMBL27795544 0.82 CHRM2 (0.47) ALDH1A1HDAC1HDAC6HDAC8HDAC3
SCHEMBL6816345 0.79 ALDH1A1 (0.47) ALDH1A1HDAC1HDAC6HDAC8HDAC3
SCHEMBL845803 0.77 ALDH1A1 (0.56) ALDH1A1HDAC1HDAC6HDAC8HDAC3
SCHEMBL28280822 0.75 ALDH1A1 (0.57) ALDH1A1HDAC1HDAC6HDAC3HDAC2
SCHEMBL20178650 0.75 ACHE (0.54) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL30041535 0.74 ALDH1A1 (0.58) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL2817935 0.74 ALDH1A1 (0.58) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL1310717 0.74 HDAC1 (0.49) ALDH1A1HDAC1HDAC6HDAC8HDAC3
SCHEMBL4929256 0.72 ALDH1A1 (0.57) ALDH1A1PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563094-A Acyclic derivatives, their preparation method and the pharmaceutical composition containing them that new (miscellaneous) aryl replaces 法国施维雅药厂 2019-04-02 CN disclosed