SCHEMBL28291608

SCHEMBL28291608

CS(=O)(=O)Nc1ccc2[nH]c(CCOC=O)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.50
MMP13 P45452 1/20 0.50
VCP P55072 3/20 0.37
MTNR1A P48039 2/20 0.36
MTNR1B P49286 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
SPR P35270 1/20 0.35
BRPF1 P55201 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ITK Q08881 1/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
OGT O15294 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28293142 0.90 MMP2 (0.40) MMP2MMP13MTNR1AMTNR1BGRIN1
SCHEMBL27521819 0.84 MTNR1A (0.36) MMP2MMP13VCPMTNR1AMTNR1B
SCHEMBL9371052 0.81 MMP2 (0.50) MMP2MMP13VCPMTNR1AMTNR1B
SCHEMBL9370958 0.79 MMP2 (0.56) MMP2MMP13VCPMTNR1AMTNR1B
SCHEMBL9371502 0.79 MMP2 (0.53) MMP2MMP13VCPMTNR1AMTNR1B
SCHEMBL27613737 0.78 LOXL2 (0.54) MTNR1AMTNR1BSMN1; SMN2LMNAKDM4E
SCHEMBL28072238 0.78 LOXL2 (0.54) MTNR1AMTNR1BSMN1; SMN2KDM4EALDH1A1
SCHEMBL9371043 0.78 MMP2 (0.52) MMP2MMP13VCPMTNR1AMTNR1B
SCHEMBL28672705 0.76 LOXL2 (0.58) MTNR1AMTNR1BSMN1; SMN2LMNAKDM4E
SCHEMBL28038688 0.76 KDM4E (0.40) MTNR1AMTNR1BSMN1; SMN2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748840-A A kind of synthetic method of 2- substituted indole derivative 中国医学科学院药物研究所 2019-05-14 CN disclosed