SCHEMBL28291778

SCHEMBL28291778

N#Cc1ccc(CCC2CCCN2CCc2ccc(C#N)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.59
KCNH2 Q12809 2/20 0.54
KCNJ1 P48048 1/20 0.54
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
SPHK2 Q9NRA0 2/20 0.47
SPHK1 Q9NYA1 2/20 0.47
SLC6A4 P31645 1/20 0.46
TRPV6 Q9H1D0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28290374 0.81 OPRK1 (0.56) HRH3SPHK2SPHK1TRPV6
SCHEMBL28290323 0.81 SPHK2 (0.50) HRH3SPHK2SPHK1TRPV6
SCHEMBL28872406 0.78 SLC18A2 (0.53) HRH3KCNH2SPHK2SPHK1
SCHEMBL28291886 0.77 MAOB (0.48) HRH3MAOBSPHK2SPHK1TRPV6
SCHEMBL28290308 0.75 HRH3 (0.70) HRH3KCNH2KCNJ1MAOASPHK2
SCHEMBL1640926 0.75 HRH3 (1.00) HRH3KCNH2SPHK2SPHK1
SCHEMBL1640070 0.75 HRH3 (1.00) HRH3KCNH2
SCHEMBL1640267 0.75 HRH3 (1.00) HRH3KCNH2SPHK2SPHK1
SCHEMBL1641177 0.75 HRH3 (1.00) HRH3KCNH2
SCHEMBL14375366 0.72 HRH3 (0.60) HRH3SPHK2SPHK1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641878-A DIPROVOCIM: a new class of effective TLR agonist 斯克里普斯研究学院 2019-04-16 CN disclosed