SCHEMBL28291873

SCHEMBL28291873

Cc1cc(N2CCN(C)CC2)c(N)cc1-c1ccc(C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.53
HSD17B10 Q99714 3/20 0.53
ALDH1A1 P00352 2/20 0.53
CHEK1 O14757 3/20 0.48
WDR5 P61964 3/20 0.47
GAA P10253 4/20 0.46
POLB P06746 4/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
NR4A1 P22736 1/20 0.45
HTR1D P28221 4/20 0.45
MAPK1 P28482 2/20 0.44
SLC6A4 P31645 2/20 0.43
TMPRSS2 O15393 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
RECQL P46063 1/20 0.43
PTK2B Q14289 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29891414 0.87 KDM4E (0.51) KDM4EHSD17B10ALDH1A1WDR5TDP1
SCHEMBL28293596 0.81 SMN1; SMN2 (0.56) ALDH1A1GAAMAPK1MAPT
SCHEMBL15776926 0.78 KDM4E (0.78) KDM4EHSD17B10ALDH1A1CHEK1WDR5
SCHEMBL17287367 0.78 KDM4E (0.60) KDM4EHSD17B10ALDH1A1CHEK1WDR5
SCHEMBL29891269 0.75 WDR5 (0.69) WDR5
SCHEMBL27968017 0.75 L3MBTL1 (0.49) KDM4EALDH1A1WDR5GAAPOLB
SCHEMBL2744322 0.75 CHEK1 (0.61) KDM4EALDH1A1CHEK1HTT
SCHEMBL29891029 0.74 WDR5 (0.52) KDM4EHSD17B10ALDH1A1WDR5L3MBTL1
SCHEMBL12752917 0.74 HSD17B10 (0.57) KDM4EHSD17B10ALDH1A1CHEK1WDR5
SCHEMBL7882534 0.73 POLB (0.57) ALDH1A1POLBL3MBTL1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-A Phenyl amines WDR5 protein-protein interaction inhibitor and its preparation method and purposes 中国药科大学 2019-05-10 CN disclosed