SCHEMBL28292382

SCHEMBL28292382

O=COCC1Cc2ccccc2C1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.43
CYP19A1 P11511 2/20 0.39
ADRA2A P08913 1/20 0.35
CHRM2 P08172 2/20 0.35
CHRM1 P11229 2/20 0.35
CHRM3 P20309 2/20 0.35
PREP P48147 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
ANPEP P15144 1/20 0.32
DRD3 P35462 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27497694 0.81 IDO1 (0.58) IDO1CYP19A1ADRA2ACHRM2CHRM1
SCHEMBL28869631 0.80 SIGMAR1 (0.46) SIGMAR1CA2
SCHEMBL27823366 0.79 PNMT (0.40) ADRA2A
SCHEMBL14439410 0.77 CHRM2 (0.35) CYP19A1CHRM2CHRM1CHRM3
Ethoxycarbonyl Group SCHEMBL27711869 0.75 IDO1 (0.37) IDO1CYP19A1CHRM2CHRM1CHRM3
SCHEMBL28294166 0.74 CA1 (0.56) CA1CA2
SCHEMBL28294086 0.74 CA1 (0.39) CA1CA2
SCHEMBL27802706 0.74 HSD17B1 (0.38) CYP19A1
SCHEMBL2741074 0.72 IDO1 (0.47) IDO1CYP19A1ADRA2ASIGMAR1ADRA1D
SCHEMBL833464 0.72 IDO1 (0.42) IDO1CYP19A1ADRA2APREPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109743875-A The inhibitor of MENIN-MLL interaction 生命医药公司 2019-05-10 CN disclosed
CN-1835753-A Spiro tetrahydroquinazolines and dihydrocyclopentapyrimidines as CFR antagonists ROCHE PALO ALTO LLC (CH) 2006-09-20 CN disclosed