SCHEMBL28292812

SCHEMBL28292812

O=C(c1cc[c]cc1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.67
AKR1C3 P42330 1/20 0.67
CYP3A4 P08684 4/20 0.62
ALDH1A1 P00352 3/20 0.62
GAA P10253 1/20 0.62
CYP2C9 P11712 3/20 0.57
CYP2C19 P33261 3/20 0.57
HSD17B10 Q99714 1/20 0.57
NAMPT P43490 2/20 0.54
CYP2D6 P10635 2/20 0.51
CYP1A2 P05177 1/20 0.51
POLB P06746 2/20 0.50
TSHR P16473 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
SLC6A7 Q99884 1/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7124360 0.84 MEN1 (0.69) ALDH1A1HSD17B10POLBTSHRMEN1
SCHEMBL7956657 0.82 SMN1; SMN2 (0.67) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA
SCHEMBL12082812 0.82 LMNA (0.69) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA
SCHEMBL6791126 0.82 SMN1; SMN2 (0.67) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA
SCHEMBL95296 0.82 SMN1; SMN2 (0.67) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA
SCHEMBL1921224 0.82 ALDH1A1 (0.56) SMN1; SMN2ALDH1A1POLBTSHRMEN1
SCHEMBL5546278 0.81 POLB (0.69) ALDH1A1HSD17B10POLBTSHRMEN1
SCHEMBL23008892 0.81 SMN1; SMN2 (0.75) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA
SCHEMBL7954884 0.81 SLC6A7 (0.63) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA
SCHEMBL5908986 0.80 SMN1; SMN2 (1.00) SMN1; SMN2AKR1C3CYP3A4ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104350055-B Bicyclic heteroaryl derivatives and application thereof as MNK1 and MNK2 regulator 新加坡科技研究局 2019-05-31 CN disclosed