SCHEMBL28293019

SCHEMBL28293019

CC(C)(C)C(=O)ON1CCN(c2ccc(Br)c(F)c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
PDK2 Q15119 2/20 0.35
MCHR1 Q99705 1/20 0.35
MAPT P10636 5/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
DRD2 P14416 2/20 0.34
DRD4 P21917 2/20 0.34
TP53 P04637 2/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TTR P02766 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MMP2 P08253 1/20 0.33
MMP13 P45452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27809025 0.86 ALKBH5 (0.41) LMNAPDK2MAPTSMN1; SMN2HTT
SCHEMBL27945026 0.86 IP6K1 (0.39) LMNAALDH1A1NR1H2NR1H3PDK2
SCHEMBL27648798 0.85 SLC6A9 (0.42) LMNAALDH1A1TSHRPDK2RORC
SCHEMBL28258173 0.85 SMN1; SMN2 (0.40) LMNAALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL27945497 0.83 IP6K1 (0.39) LMNAALDH1A1PDK2MAPTSMN1; SMN2
SCHEMBL27859336 0.82 DRD2 (0.48) LMNAALDH1A1MAPTSMN1; SMN2DRD2
SCHEMBL28808789 0.81 HDAC3 (0.32) LMNAALDH1A1NR1H2NR1H3MAPT
SCHEMBL2386743 0.81 MAPT (0.55) LMNAALDH1A1TSHRPDK2MAPT
SCHEMBL29373833 0.81 MAPT (0.55) LMNAALDH1A1TSHRPDK2MAPT
SCHEMBL27824902 0.80 ADAMTS5 (0.42) LMNAALDH1A1NR1H2NR1H3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641871-A AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS 诺华股份有限公司 2019-04-16 CN disclosed