SCHEMBL28293514

SCHEMBL28293514

CCCCC(CCCN(C)Cc1cccc2ccccc12)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.51
KMT2A Q03164 2/20 0.45
METAP2 P50579 3/20 0.44
TDP1 Q9NUW8 1/20 0.43
NR1I2 O75469 2/20 0.43
SLC6A2 P23975 2/20 0.43
HTR2A P28223 2/20 0.43
SLC6A4 P31645 2/20 0.43
KCNH2 Q12809 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
LMNA P02545 2/20 0.43
HIF1A Q16665 2/20 0.43
DRD2 P14416 1/20 0.43
ADRA2C P18825 1/20 0.43
CNR1 P21554 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRK1 P41145 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28293585 0.87 KDM4E (0.44) CYP2D6CYP1A2CYP2C19METAP2TDP1
SCHEMBL16256972 0.82 CYP2D6 (0.71) CYP2D6CYP1A2CYP2C19KMT2ANR1I2
SCHEMBL28295494 0.79 SIGMAR1 (0.48) KMT2ASIGMAR1ACHEMEN1MMP2
SCHEMBL11932504 0.78 CYP2D6 (0.65) CYP2D6CYP1A2CYP2C19KMT2AMETAP2
SCHEMBL11887346 0.77 CYP2D6 (0.79) CYP2D6CYP1A2CYP2C19KMT2ATDP1
SCHEMBL14542581 0.76 CYP2D6 (0.76) CYP2D6CYP1A2CYP2C19KMT2ATDP1
SCHEMBL28295290 0.74 TMEM97 (0.50) KMT2ASIGMAR1ACHEMEN1TSHR
SCHEMBL28049380 0.73 CYP2D6 (0.61) CYP2D6CYP1A2CYP2C19KMT2ATDP1
Hydrochloric Acid SCHEMBL5010879 0.73 DNM1 (0.51) CYP2D6CYP1A2CYP2C19HIF1ADRD2
SCHEMBL28295287 0.73 TMEM97 (0.48) SIGMAR1HTTMMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110123820-A Arginase inhibitor and its application method 阿斯利康公司 2019-08-16 CN disclosed
CN-104857005-B Arginase inhibitor and its application method 阿斯利康公司 2019-04-26 CN disclosed