SCHEMBL28294180

SCHEMBL28294180

COc1cccc(-c2ccc3nc[nH]c3c2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.69
QPCT Q16769 9/20 0.58
QPCTL Q9NXS2 8/20 0.58
MAP4K4 O95819 1/20 0.51
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.49
USP2 O75604 2/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C19 P33261 2/20 0.49
CLK4 Q9HAZ1 2/20 0.49
GLA P06280 1/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
HIF1A Q16665 1/20 0.49
CYP2C9 P11712 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2096521 0.88 MMP12 (0.55) MMP12QPCTQPCTLMAP4K4USP2
SCHEMBL2093317 0.86 MMP12 (0.75) MMP12QPCTQPCTLALDH1A1
SCHEMBL225932 0.82 MMP12 (1.00) MMP12QPCTQPCTLPOLBMAPT
SCHEMBL29424791 0.82 MMP12 (1.00) MMP12QPCTQPCTLPOLBMAPT
SCHEMBL8634290 0.80 QPCT (0.68) MMP12QPCTQPCTLMAPTALDH1A1
SCHEMBL13680531 0.80 QPCT (0.60) MMP12QPCTQPCTLMAP4K4MAPT
SCHEMBL22418756 0.79 QPCT (0.64) QPCTQPCTLMAPTALDH1A1
SCHEMBL2462345 0.79 QPCT (0.68) QPCTQPCTLMAPTALDH1A1
Benzimidazole SCHEMBL15413095 0.78 MMP12 (0.84) MMP12QPCTQPCTLPOLBALDH1A1
SCHEMBL23227938 0.76 QPCT (0.60) QPCTQPCTLMAP4K4MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107312008-B A kind of catalysis prepares the catalyst and system and method for benzimidazole simultaneously [2,1-b] quinoline -6- ketone derivatives 马鞍山市泰博化工科技有限公司 2019-08-27 CN disclosed
CN-106866543-B A method of benzimidazole compound is catalyzed and synthesized under microwave radiation in water phase 福建医科大学 2019-05-14 CN disclosed
CN-107312008-A A kind of easy catalysis prepares the catalyst and system and method for benzimidazole simultaneously ketone derivatives of [2,1 b] quinoline 6 马鞍山市泰博化工科技有限公司 2017-11-03 CN disclosed