SCHEMBL28294570

SCHEMBL28294570

CCc1oc2cccc(Br)c2c1-c1ccc(O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 5/20 0.48
PTPN1 P18031 4/20 0.46
SLC22A12 Q96S37 6/20 0.42
EYA3 Q99504 5/20 0.42
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
ESR1 P03372 3/20 0.39
PPARG P37231 2/20 0.39
EYA2 O00167 1/20 0.39
MEN1 O00255 1/20 0.39
ABCC4 O15439 1/20 0.39
PLIN1 O60240 1/20 0.39
NR1I2 O75469 1/20 0.39
USP2 O75604 1/20 0.39
ABCB11 O95342 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
ALB P02768 1/20 0.39
NR3C1 P04150 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28104534 0.77 SLC22A12 (0.40) TTRPTPN1SLC22A12EYA3CYP2C9
SCHEMBL7499188 0.76 PTPN1 (0.74) TTRPTPN1SLC22A12EYA3CYP2C9
SCHEMBL28249620 0.74 MAPT (0.45) TTRPTPN1SLC22A12EYA3ESR1
SCHEMBL28061856 0.71 GABRA1 (0.45) ESR1MEN1KMT2AESR2
SCHEMBL27498982 0.69 ESR1 (0.48) ESR1MEN1USP2ALDH1A1LMNA
SCHEMBL5483047 0.69 MEN1 (0.41) TTRPTPN1SLC22A12EYA3CYP2C9
SCHEMBL28220577 0.69 SLC22A12 (0.56) TTRPTPN1SLC22A12EYA3CYP2C9
SCHEMBL28104532 0.67 CYP2C19 (0.62) TTRPTPN1SLC22A12EYA3CYP2C9
SCHEMBL23532166 0.65 TTR (0.42) TTRPTPN1SLC22A12EYA3CYP2C9
SCHEMBL28282749 0.65 USP7 (0.43) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105218479-B The new derivatives, preparation method and application of 2- [3- cyano-4-isobutoxy phenyl] -4- methylthiazol-5-formic acid 湘北威尔曼制药股份有限公司 2019-10-25 CN disclosed
CN-105272984-B Pyrazolo [3,4-d] pyrimidin-4-one-derivatives, preparation method and application 湘北威尔曼制药股份有限公司 2019-06-14 CN disclosed
CN-106470981-B The new derivatives, preparation method and application of 2- [3- cyano-4-isobutoxy phenyl] -4- methylthiazol-5-formic acid 湘北威尔曼制药股份有限公司 2019-05-07 CN disclosed