SCHEMBL28294626

SCHEMBL28294626

Cc1nc(N)c2cc(Cc3cccc(Cl)c3)ccc2n1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
HIF1A Q16665 1/20 0.48
PNMT P11086 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR6 P50406 1/20 0.41
PDE5A O76074 1/20 0.40
CCR2 P41597 1/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294625 0.81 NR4A2 (0.52) APPKDM4ECYP3A4CYP2C19HIF1A
SCHEMBL25722168 0.76 ALDH1A1 (0.51) KDM4EHTTSMN1; SMN2
SCHEMBL18895408 0.76 DHFR (0.42) APPPNMTHTTSMN1; SMN2CCR2
SCHEMBL18895154 0.74 HTT (0.54) APPKDM4ECYP3A4CYP2C19HTT
SCHEMBL5354603 0.73 HSP90AB1 (0.51) KDM4ECYP3A4CYP2C19HIF1A
SCHEMBL28957472 0.72 NR4A2 (0.62) APPPNMTNOS3NOS1MAP4K4
SCHEMBL8886921 0.72 APP (0.64) APPHTR6PDE5A
SCHEMBL5355383 0.72 DHFR (0.60)
Hydrochloric Acid SCHEMBL8500111 0.71 APP (0.62) APPKDM4EHTR6PDE5A
SCHEMBL3300276 0.70 PNMT (0.65) CYP3A4PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641886-A bicyclic BET bromodomain inhibitors and uses thereof 康威基内有限公司 2019-04-16 CN disclosed