SCHEMBL28294625

SCHEMBL28294625

Cc1cc(N)c2cc(Cc3cccc(Cl)c3)ccc2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.52
NCF1 P14598 1/20 0.49
ALDH1A1 P00352 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
HIF1A Q16665 1/20 0.48
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
HCRTR1 O43613 1/20 0.46
OPRL1 P41146 2/20 0.45
TERT O14746 2/20 0.44
GNG2 P59768 2/20 0.43
GNB1 P62873 2/20 0.43
MMP1 P03956 1/20 0.43
MMP9 P14780 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294626 0.81 APP (0.48) KDM4ECYP3A4CYP2C19HIF1AAPP
SCHEMBL8242755 0.80 ALDH1A1 (0.49) NR4A2NCF1ALDH1A1CASP1CASP7
SCHEMBL440491 0.79 NR4A2 (0.74) NR4A2NCF1ALDH1A1CASP1CASP7
SCHEMBL13039504 0.78 ALDH1A1 (0.50) NR4A2NCF1ALDH1A1CASP1CASP7
SCHEMBL28957472 0.78 NR4A2 (0.62) NR4A2NCF1APP
SCHEMBL439542 0.76 ALDH1A1 (0.58) NR4A2NCF1ALDH1A1CASP1CASP7
SCHEMBL3300276 0.70 PNMT (0.65) CYP3A4
SCHEMBL18586524 0.70 MPO (0.55) CYP3A4KMT2AMEN1USP2
SCHEMBL438119 0.70 NR4A2 (1.00) NR4A2NCF1ALDH1A1CASP1CASP7
SCHEMBL21384185 0.69 TAAR1 (0.57) ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109641886-A bicyclic BET bromodomain inhibitors and uses thereof 康威基内有限公司 2019-04-16 CN disclosed