SCHEMBL28295474

SCHEMBL28295474

CC1CNc2ccccc2C(c2ccccc2)=N1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 5/20 0.56
CCKBR P32239 4/20 0.49
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
GABRA1 P14867 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
GABRA2 P47869 2/20 0.43
GABRB2 P47870 2/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
CCKAR P32238 2/20 0.39
HDAC1 Q13547 1/20 0.39
CCNE2 O96020 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
BACE1 P56817 1/20 0.38
NOS2 P35228 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297188 0.83 CHRM1 (0.49) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL11684302 0.82 CHRM1 (0.62) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL29695279 0.82 CCKBR (0.48) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL6065137 0.82 CCKBR (0.48) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL27675515 0.82 CCKBR (0.48) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL28297197 0.78 LMNA (0.57) CHRM1MEN1KMT2AGABRA1GABRA5
SCHEMBL20226281 0.77 CHRM1 (0.61) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL20098126 0.75 CCKBR (0.46) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL20226277 0.75 CHRM1 (0.58) CHRM1CCKBRMEN1ALDH1A1KMT2A
SCHEMBL11278574 0.73 GABRA1 (0.47) CHRM1CCKBRMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN claimed
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN disclosed