SCHEMBL28295982

SCHEMBL28295982

Cc1cc(Br)c([N+](=O)[O-])c(N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
LMNA P02545 4/20 0.46
HTT P42858 4/20 0.46
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
TDP1 Q9NUW8 3/20 0.39
KMT2A Q03164 2/20 0.39
MITF O75030 1/20 0.39
MGMT P16455 1/20 0.38
ALDH1A1 P00352 4/20 0.38
CYP3A4 P08684 2/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31056280 0.81 MAPT (0.48) MAPTLMNAHTTRAB9ANPC1
SCHEMBL8884172 0.81 GRIN2D (0.41) MAPTLMNAHTTGRIN2DGRIN3B
SCHEMBL4522152 0.81 GRIN2D (0.41) MAPTLMNAHTTRAB9ANPC1
SCHEMBL31128165 0.81 GRIN2D (0.41) MAPTLMNAHTTRAB9ANPC1
SCHEMBL7385881 0.81 MAPT (0.48) MAPTLMNAHTTRAB9ANPC1
SCHEMBL803098 0.79 ALDH1A1 (0.47) MAPTLMNAHTTRAB9ANPC1
SCHEMBL28720365 0.79 GRIN2D (0.40) MAPTLMNAHTTGRIN2DGRIN3B
SCHEMBL2322399 0.74 GRIN2D (0.49) MAPTLMNAHTTGRIN2DGRIN3B
SCHEMBL9721947 0.72 NOS3 (0.55) MAPTLMNAHTTRAB9ANPC1
SCHEMBL26694656 0.72 KDM4E (0.42) MAPTLMNAHTTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-A Inhibitor as PARP1, PARP2 and/or tubulin can be used for the phthalazine derivatives for the treatment of cancer 加利福尼亚大学董事会 2019-06-04 CN disclosed