SCHEMBL28296320

SCHEMBL28296320

COc1ccc(/C=C/c2ccccc2/C(N)=N/c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.53
RELA Q04206 3/20 0.51
NFE2L2 Q16236 2/20 0.51
SNCA P37840 5/20 0.47
KDM4E B2RXH2 2/20 0.45
CYP1A1 P04798 2/20 0.45
CYP1B1 Q16678 2/20 0.45
LMNA P02545 1/20 0.45
ALOX12 P18054 1/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
PLG P00747 1/20 0.44
PLAU P00749 1/20 0.44
PLAT P00750 1/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NOS3 P29474 2/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28410291 1.00 TRPA1 (0.53) TRPA1RELANFE2L2SNCAKDM4E
SCHEMBL28410290 1.00 TRPA1 (0.53) TRPA1RELANFE2L2SNCAKDM4E
SCHEMBL28408256 0.85 MEN1 (0.48) TRPA1NFE2L2LMNAPLAUPLAT
SCHEMBL28408254 0.85 MEN1 (0.48) TRPA1NFE2L2LMNAPLAUPLAT
SCHEMBL28408255 0.85 MEN1 (0.48) TRPA1NFE2L2LMNAPLAUPLAT
SCHEMBL28410294 0.82 NFE2L2 (0.50) TRPA1NFE2L2SNCALMNAPTGS1
SCHEMBL28410295 0.82 NFE2L2 (0.50) TRPA1NFE2L2SNCALMNAPTGS1
SCHEMBL28296333 0.82 NFE2L2 (0.50) TRPA1NFE2L2SNCALMNAPTGS1
SCHEMBL5335032 0.79 TRPA1 (0.61) TRPA1RELANFE2L2SNCAKDM4E
SCHEMBL5335033 0.79 TRPA1 (0.61) TRPA1RELANFE2L2SNCAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796372-B Method for preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2020-03-10 CN disclosed
CN-109796372-A A method of preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2019-05-24 CN disclosed