SCHEMBL28296333

SCHEMBL28296333

N/C(=N\c1ccccc1)c1ccccc1/C=C/c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 7/20 0.50
SNCA P37840 2/20 0.44
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PTGS1 P23219 1/20 0.40
SLC22A2 O15244 2/20 0.40
SLC22A1 O15245 2/20 0.40
SLC22A3 O75751 2/20 0.40
PLAU P00749 2/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
EGFR P00533 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28410295 1.00 NFE2L2 (0.50) NFE2L2SNCAGRIN1GRIN2BMEN1
SCHEMBL28410294 1.00 NFE2L2 (0.50) NFE2L2SNCAGRIN1GRIN2BMEN1
SCHEMBL28408255 0.89 MEN1 (0.48) NFE2L2MEN1KMT2ASLC22A2SLC22A1
SCHEMBL28408254 0.89 MEN1 (0.48) NFE2L2MEN1KMT2ASLC22A2SLC22A1
SCHEMBL28408256 0.89 MEN1 (0.48) NFE2L2MEN1KMT2ASLC22A2SLC22A1
SCHEMBL28410290 0.82 TRPA1 (0.53) NFE2L2SNCAPTGS1PLAUEGFR
SCHEMBL28410291 0.82 TRPA1 (0.53) NFE2L2SNCAPTGS1PLAUEGFR
SCHEMBL28296320 0.82 TRPA1 (0.53) NFE2L2SNCAPTGS1PLAUEGFR
SCHEMBL9797944 0.76 NFE2L2 (0.58) NFE2L2SNCAMAOAMAOBALDH1A1
SCHEMBL10496469 0.76 NFE2L2 (0.58) NFE2L2SNCAMAOAMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796372-B Method for preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2020-03-10 CN disclosed
CN-109796372-A A method of preparing polysubstituted alkenyl amidine 中国科学院化学研究所 2019-05-24 CN disclosed