SCHEMBL28296473

SCHEMBL28296473

O=COC(=O)C1CCNC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 4/20 0.40
GABRB2 P47870 3/20 0.40
TSHR P16473 3/20 0.40
GABRA1 P14867 3/20 0.40
GABRA4 P48169 2/20 0.40
GABRG2 P18507 2/20 0.40
GABRB3 P28472 2/20 0.40
GABRA3 P34903 2/20 0.40
GABRA2 P47869 2/20 0.40
GABRA6 Q16445 2/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRE P78334 1/20 0.40
PMP22 Q01453 1/20 0.40
GABRG1 Q8N1C3 1/20 0.40
GABRG3 Q99928 1/20 0.40
GABRQ Q9UN88 1/20 0.40
SLC6A1 P30531 4/20 0.39
SLC6A11 P48066 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27991990 0.88 GABRA5 (0.48) GABRA5GABRB2TSHRGABRA1GABRA4
SCHEMBL9212263 0.82 GABRA5 (0.39) GABRA5GABRB2TSHRGABRA1GABRA4
SCHEMBL16114958 0.76 GABRA5 (0.40) GABRA5GABRB2TSHRGABRA1GABRA4
SCHEMBL31249843 0.76 SLC6A1 (0.39) GABRA5GABRB2TSHRGABRA1GABRA4
SCHEMBL11239979 0.75
SCHEMBL6939540 0.75 ELANE (0.34) SMN1; SMN2KMT2A
SCHEMBL10703008 0.75
SCHEMBL1161879 0.75
SCHEMBL12699753 0.75
SCHEMBL584094 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207515-B Pyrazine compounds for the treatment of infectious diseases 豪夫迈·罗氏有限公司 2019-05-28 CN disclosed