SCHEMBL27991990

SCHEMBL27991990

O=COC(=O)C1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 4/20 0.48
GABRA1 P14867 3/20 0.48
GABRB2 P47870 3/20 0.48
TSHR P16473 2/20 0.48
GABRG2 P18507 2/20 0.48
GABRB3 P28472 2/20 0.48
GABRA3 P34903 2/20 0.48
GABRA2 P47869 2/20 0.48
GABRA6 Q16445 2/20 0.48
GABRA4 P48169 2/20 0.48
GABRP O00591 1/20 0.48
GABRD O14764 1/20 0.48
GABRB1 P18505 1/20 0.48
GABRE P78334 1/20 0.48
PMP22 Q01453 1/20 0.48
GABRG1 Q8N1C3 1/20 0.48
GABRG3 Q99928 1/20 0.48
GABRQ Q9UN88 1/20 0.48
LMNA P02545 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28296473 0.88 GABRA5 (0.40) GABRA5GABRA1GABRB2TSHRGABRG2
SCHEMBL11239979 0.84
SCHEMBL6939540 0.84 ELANE (0.34) MEN1KMT2ASMN1; SMN2
SCHEMBL13675135 0.79
SCHEMBL27530748 0.79 CES2 (0.42) TSHRPOLBKMT2AALDH1A1SMN1; SMN2
SCHEMBL14763815 0.77 CES2 (0.46) TSHRPOLBKMT2AALDH1A1SMN1; SMN2
SCHEMBL6881837 0.77 CES2 (0.46) TSHRPOLBKMT2AALDH1A1SMN1; SMN2
SCHEMBL3997244 0.77 GABRA1 (0.56) GABRA5GABRA1GABRB2TSHRGABRG2
SCHEMBL9205374 0.76 GABRP (0.42) GABRA5GABRA1GABRB2TSHRGABRG2
SCHEMBL27755064 0.76 LMNA (0.40) GABRA5GABRA1GABRB2TSHRGABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115485279-A Antibacterial 8-phenylamino-3- (pyrazol-4-yl) imidazo [1,2-a ] pyrazine derivatives 豪夫迈·罗氏有限公司 2022-12-16 CN claimed
CN-115485279-A Antibacterial 8-phenylamino-3- (pyrazol-4-yl) imidazo [1,2-a ] pyrazine derivatives 豪夫迈·罗氏有限公司 2022-12-16 CN disclosed
CN-110041335-A It is a kind of to improve the water-soluble method of couroupitine A, tryptamines ketone derivatives and its preparation method and application 同济大学 2019-07-23 CN disclosed
CN-104211635-A Piperidine compounds, and preparation method, pharmaceutical compositions and use thereof SHANGHAI INST MATERIA MEDICA 2014-12-17 CN disclosed