SCHEMBL28296852

SCHEMBL28296852

Fc1cc(F)c(F)c(C2CCNC2)c1F.NC=S

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.38
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
CYP2D6 P10635 1/20 0.35
DPP4 P27487 1/20 0.35
MPO P05164 1/20 0.34
HTR2C P28335 2/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28298510 0.90 SLC6A2 (0.40) HTR3ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL19995575 0.90 SLC6A2 (0.40) HTR3ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL28296879 0.86 HTR3A (0.38) HTR3AMPOHTR2C
SCHEMBL28296843 0.84 HTR3A (0.38) HTR3ASLC6A2SLC6A4SLC6A3MPO
SCHEMBL28296873 0.81 CHRNB2 (0.44) HTR3ASLC6A2SLC6A4SLC6A3DPP4
SCHEMBL28873499 0.80 HCAR2 (0.38) HTR3AMPOHTR2CCHRNB2CHRNB4
SCHEMBL28873365 0.77 HTR3A (0.43) HTR3ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL28298499 0.77 HTR3A (0.43) HTR3ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL28296838 0.77 HTR3A (0.43) HTR3ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL28298496 0.76 HTR3A (0.51) HTR3ASLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed