SCHEMBL28296879

SCHEMBL28296879

Fc1c(F)c(F)c(C2CCNC2)c(F)c1F.NC=S

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.38
HTR2C P28335 2/20 0.33
MPO P05164 1/20 0.31
SLC18A3 Q16572 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19996154 0.88 HTR3A (0.41) HTR3AHTR2CMPO
SCHEMBL28296852 0.86 HTR3A (0.38) HTR3AHTR2CMPO
SCHEMBL28296843 0.80 HTR3A (0.38) HTR3AHTR2CMPO
SCHEMBL5542721 0.75 HTR1A (0.42) HTR2CSLC18A3SIGMAR1
SCHEMBL28298501 0.75 HTR3A (0.56) HTR3AHTR2CMPO
SCHEMBL28873365 0.75 HTR3A (0.43) HTR3AHTR2CMPO
SCHEMBL28298499 0.75 HTR3A (0.43) HTR3AHTR2CMPO
SCHEMBL28296838 0.75 HTR3A (0.43) HTR3AHTR2CMPO
SCHEMBL28296881 0.74 HTR3A (0.42) HTR3AHTR2C
SCHEMBL19995575 0.73 SLC6A2 (0.40) HTR3AHTR2CMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed