SCHEMBL28297780

SCHEMBL28297780

CCOC(=O)C(C(=O)OCC)[C@@H](Cc1cc(F)cc(F)c1)[N+](=O)[O-]

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 7/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
FBP1 P09467 1/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
MAPK1 P28482 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
EPHX2 P34913 1/20 0.33
PPARG P37231 1/20 0.33
ALDH1A1 P00352 6/20 0.33
NR3C1 P04150 1/20 0.33
PGR P06401 1/20 0.33
NR3C2 P08235 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28331075 0.80 MMP8 (0.50) NPC1SMN1; SMN2EPHX2PPARGALDH1A1
SCHEMBL27829606 0.80 MMP8 (0.50) NPC1SMN1; SMN2EPHX2PPARGALDH1A1
SCHEMBL28332593 0.78 MME (0.40) NPC1KMT2AMEN1MAPTCRHBP
SCHEMBL28297783 0.76 MAPT (0.36) KMT2AMEN1MAPTCRHBPCRHR2
SCHEMBL23455090 0.72 ALDH1A1 (0.48) NPC1KMT2AMEN1MAPTCRHBP
SCHEMBL21527887 0.72 ALDH1A1 (0.48) NPC1KMT2AMEN1MAPTCRHBP
SCHEMBL21527885 0.72 ALDH1A1 (0.48) NPC1KMT2AMEN1MAPTCRHBP
SCHEMBL15261624 0.71 MMP8 (0.42) KMT2AMEN1L3MBTL1SMN1; SMN2MAPK1
SCHEMBL20002387 0.70 SMN1; SMN2 (0.44) KMT2AMEN1L3MBTL1SMN1; SMN2MAPK1
SCHEMBL19996010 0.69 MAPT (0.37) NPC1KMT2AMEN1MAPTCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715633-A Dopamine-B-hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed