SCHEMBL28299458

SCHEMBL28299458

N#Cc1c[c]c([N+](=O)[O-])cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 5/20 0.47
MAPT P10636 4/20 0.38
GRIA1 P42261 2/20 0.38
GRIA2 P42262 2/20 0.38
GRIA3 P42263 2/20 0.38
GRIA4 P48058 2/20 0.38
GRM6 O15303 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALOX15 P16050 1/20 0.38
POLB P06746 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
APEX1 P27695 1/20 0.37
BLM P54132 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2208121 0.77 HSD17B10 (0.42) VCAM1TDP1GRIN2DGRIN3BGRIN1
SCHEMBL1898245 0.76 GRIN2D (0.39) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL27684781 0.73 ALDH1A1 (0.36) VCAM1MAPTALOX15HPGDTDP1
SCHEMBL9653201 0.73 ALDH1A1 (0.36) CYP1A2TDP1GRIN2DGRIN3BGRIN1
SCHEMBL1895507 0.72 ALDH1A1 (0.40) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL6282528 0.71 TSHR (0.42) VCAM1ALOX15HPGDTDP1ALDH1A1
SCHEMBL11329936 0.71 VCAM1 (0.62) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL28774035 0.69 ALDH1A1 (0.36) VCAM1MAPTALOX15HPGDTDP1
SCHEMBL1343713 0.69 VCAM1 (0.61) VCAM1MAPTGRIA1GRIA2GRIA3
SCHEMBL1624405 0.69 VCAM1 (0.56) VCAM1MAPTGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105622580-B Benzimidazole as prolyl hydroxylase inhibitors 詹森药业有限公司 2019-06-21 CN disclosed