SCHEMBL28300293

SCHEMBL28300293

COc1ccc(-c2cncnc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.52
KDM4E B2RXH2 3/20 0.50
TP53 P04637 2/20 0.50
ATM Q13315 1/20 0.50
MAPT P10636 1/20 0.50
MAP4K4 O95819 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CYP11B1 P15538 4/20 0.47
CYP11B2 P19099 4/20 0.47
CYP17A1 P05093 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
USP2 O75604 1/20 0.47
CYP2C9 P11712 1/20 0.47
NPC1 O15118 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alcohol SCHEMBL28257149 0.90 LMNA (0.49) ESR2KDM4ETP53ATMMAPT
SCHEMBL4509505 0.82 CYP11B2 (0.72) CYP11B1CYP11B2CYP17A1CYP1A2CYP3A4
SCHEMBL197522 0.80 CA1 (0.79) ESR2KDM4ETP53MAPTCA12
SCHEMBL6733562 0.80 CA1 (0.79) ESR2KDM4ETP53MAPTCA12
SCHEMBL6682176 0.80 ATM (0.72) KDM4ETP53ATMMAPTCYP1A2
SCHEMBL9151672 0.80 CA1 (0.79) ESR2KDM4ETP53MAPTCA12
SCHEMBL21960161 0.78 CYP11B1 (0.73) MAP4K4CYP11B1CYP11B2CYP17A1CYP1A2
SCHEMBL11396596 0.77 LTA4H (0.54) KDM4ETP53MAPTCA12CA1
SCHEMBL21345911 0.77 NPSR1 (0.53) ATMMAPTCYP2C9NPC1RAB9A
SCHEMBL22778252 0.77 CYP11B2 (0.72) KDM4EMAPTCYP11B1CYP11B2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232025-A1 PHOSPHINE REAGENTS FOR AZINE FLUOROALKYLATION COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2023-08-30 EP disclosed
WO-2022087129-A9 PHOSPHINE REAGENTS FOR AZINE FLUOROALKYLATION COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2022-05-27 WO disclosed
WO-2022087129-A1 PHOSPHINE REAGENTS FOR AZINE FLUOROALKYLATION COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2022-04-28 WO disclosed
CN-107207516-B Octahydro pyrrolo- [3,4-c] azole derivatives and application thereof 广东东阳光药业有限公司 2019-06-25 CN disclosed
CN-102014900-B Method of treating cancer using a neuropeptide Y5R (NPY5R) antagonist UNIV HEALTH NETWORK 2014-04-02 CN disclosed
CN-102014900-A Method of treating cancer using a neuropeptide Y5R (NPY5R) antagonist UNIV HEALTH NETWORK 2011-04-13 CN disclosed