SCHEMBL28303166

SCHEMBL28303166

CCc1c2ccc-2c1N.O=C(O)c1cncnc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 3/20 0.35
GABRD O14764 3/20 0.35
GABRA1 P14867 3/20 0.35
GABRB1 P18505 3/20 0.35
GABRG2 P18507 3/20 0.35
GABRB3 P28472 3/20 0.35
GABRA5 P31644 3/20 0.35
GABRA3 P34903 3/20 0.35
GABRA2 P47869 3/20 0.35
GABRB2 P47870 3/20 0.35
GABRA4 P48169 3/20 0.35
GABRE P78334 3/20 0.35
GABRA6 Q16445 3/20 0.35
GABRG1 Q8N1C3 3/20 0.35
GABRG3 Q99928 3/20 0.35
GABRQ Q9UN88 3/20 0.35
KDM4E B2RXH2 5/20 0.35
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
SYK P43405 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671209 0.79 ASPH (0.43) KDM4EITGB1ITGA4SYKHSD17B10
Trimethylammonium SCHEMBL8541657 0.75 ASPH (0.38) KDM4EITGB1ITGA4SYKHSD17B10
Trimethylammonium SCHEMBL8543218 0.75 ASPH (0.38) KDM4EITGB1ITGA4SYKHSD17B10
3-Chloroaniline SCHEMBL27676204 0.70 ALDH1A1 (0.41) ITGB1ITGA4SYKALDH1A1
SCHEMBL23631773 0.68 SYK (0.48) KDM4EITGB1ITGA4SYKKMT2A
SCHEMBL8574991 0.68 NFKB1 (0.40) KDM4EITGB1ITGA4SYKHSD17B10
SCHEMBL6775372 0.67 KDM4E (0.62) KDM4EKMT2AALDH1A1HPGDTSHR
SCHEMBL1012918 0.67 HCAR2 (0.39) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL13531248 0.65 KDM4E (0.49) KDM4EALDH1A1MGLLTDP1CYP3A4
SCHEMBL16592100 0.65 VNN1 (0.38) KDM4EHSD17B10ALDH1A1TDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106831603-B A kind of preparation method containing fluoropyrimidine compound 辽宁大学 2019-07-02 CN disclosed
CN-106831603-A A kind of preparation method containing fluoropyrimidine compound 辽宁大学 2017-06-13 CN disclosed