SCHEMBL28304239

SCHEMBL28304239

CC(C)(C)OC(=O)N1CCNCC1c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.50
NR1H3 Q13133 4/20 0.50
PARP1 P09874 1/20 0.43
RORC P51449 2/20 0.42
KMT2A Q03164 1/20 0.40
PDE5A O76074 1/20 0.37
DPP4 P27487 1/20 0.37
DPP7 Q9UHL4 1/20 0.37
USP30 Q70CQ3 1/20 0.36
UCHL1 P09936 1/20 0.36
FPR2 P25090 3/20 0.36
FPR3 P25089 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3697218 0.89 DPP4 (0.47) NR1H2NR1H3PARP1RORCKMT2A
SCHEMBL25913721 0.89 DPP4 (0.47) NR1H2NR1H3PARP1RORCKMT2A
SCHEMBL8140446 0.88 PARP1 (0.43) NR1H2NR1H3PARP1DPP4DPP7
SCHEMBL1673503 0.88 MEN1 (0.43) NR1H2NR1H3PARP1KMT2A
SCHEMBL4325057 0.87 NR1H2 (0.49) NR1H2NR1H3PARP1RORCDPP4
SCHEMBL22285173 0.87 NR1H2 (0.49) NR1H2NR1H3PARP1RORCDPP4
SCHEMBL874416 0.87 NR1H2 (0.49) NR1H2NR1H3PARP1RORCDPP4
SCHEMBL31470897 0.85 GPR119 (0.46) NR1H2NR1H3PARP1
SCHEMBL31408651 0.85 PARP1 (0.41) NR1H2NR1H3PARP1KMT2ADPP4
SCHEMBL8880888 0.85 GPR119 (0.46) NR1H2NR1H3PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178377-A Pain-resistant compounds and methods of making the same 山东新时代药业有限公司 2023-05-30 CN disclosed
CN-111417637-B Anti-pain compounds and process for preparing same 山东新时代药业有限公司 2022-09-13 CN disclosed
CN-109897044-A Anti- neurogenic pain compound and preparation method thereof 北京大学 2019-06-18 CN disclosed