SCHEMBL28306404

SCHEMBL28306404

COc1ccc(Sc2cc(CN)ccc2N2CCNCC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 16/20 0.63
HTR1A P08908 15/20 0.63
HTR2C P28335 2/20 0.51
HTR3E A5X5Y0 2/20 0.49
HTR3B O95264 2/20 0.49
HTR3D Q70Z44 2/20 0.49
HTR3C Q8WXA8 2/20 0.49
CYP1A2 P05177 4/20 0.46
CYP3A4 P08684 4/20 0.46
CYP2D6 P10635 4/20 0.46
CYP2C9 P11712 4/20 0.46
HTR6 P50406 1/20 0.46
ADRB1 P08588 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
HTR7 P34969 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28231884 0.91 HTR3A (0.71) HTR3AHTR1AHTR2CHTR3EHTR3B
SCHEMBL546686 0.83 HTR3A (0.81) HTR3AHTR1AHTR2CHTR3EHTR3B
SCHEMBL546581 0.82 HTR3A (0.67) HTR3AHTR1AHTR2CHTR3EHTR3B
SCHEMBL27550397 0.76 HTR1A (0.71) HTR3AHTR1ACYP1A2CYP3A4CYP2D6
SCHEMBL546511 0.76 HTR3A (1.00) HTR3AHTR1AHTR2CHTR3EHTR3B
Tert-Butyl Formate SCHEMBL28112175 0.76 HTR1A (0.43) HTR3AHTR1AHTR2CCYP1A2CYP3A4
SCHEMBL27568938 0.75 HTR1A (0.67) HTR3AHTR1ACYP1A2CYP3A4CYP2D6
SCHEMBL17260217 0.73 HTR3E (0.62) HTR3AHTR1AHTR2CHTR3EHTR3B
SCHEMBL28254187 0.72 HTR3A (0.71) HTR3AHTR1AHTR2CHTR3EHTR3B
SCHEMBL547373 0.72 HTR3A (0.71) HTR3AHTR1AHTR2CHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110022869-A For skin and/or the serotonin 1B receptor stimulators of hair reparation 巴斯德研究院 2019-07-16 CN disclosed
CN-108348486-A 5-hydroxytryptamine 1B receptor agonists as promoters for satellite cell self-renewal and/or differentiation 巴斯德研究院 2018-07-31 CN disclosed