SCHEMBL28308671

SCHEMBL28308671

C=Cc1nccc(-c2ccccc2)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.42
PDCD1 Q15116 3/20 0.40
CD274 Q9NZQ7 3/20 0.40
GRM4 Q14833 1/20 0.39
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
DAPK3 O43293 1/20 0.39
JAK2 O60674 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
PAK4 O96013 1/20 0.39
CSF1R P07333 1/20 0.39
RET P07949 1/20 0.39
IGF1R P08069 1/20 0.39
FGFR1 P11362 1/20 0.39
PRKACA P17612 1/20 0.39
FLT1 P17948 1/20 0.39
LTK P29376 1/20 0.39
GRK5 P34947 1/20 0.39
KDR P35968 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL554430 0.81 LRRK2 (0.39) CHEK1IKBKBCHUKDAPK3JAK2
SCHEMBL28309533 0.77 POLB (0.40) LRRK2BTKALDH1A1KMT2APTGS1
SCHEMBL10824239 0.77 TOP1 (0.40) ALDH1A1PTGS1PTGS2MAPT
SCHEMBL10199428 0.76 GRM4 (0.58) CHEK1PDCD1CD274GRM4IKBKB
SCHEMBL28309538 0.76 IKBKB (0.35) CHEK1IKBKBCHUKDAPK3JAK2
SCHEMBL2977681 0.76 ALDH1A1 (0.55) LRRK2CYP1A2MEN1ALDH1A1KMT2A
Iodide SCHEMBL27658785 0.76 TOP1 (0.39) BTKALDH1A1PTGS1PTGS2MAPT
SCHEMBL15865503 0.75 NOS3 (0.54) CHEK1PDCD1CD274GRM4IKBKB
SCHEMBL11606622 0.75 CHEK1 (0.46) CHEK1PDCD1CD274GRM4IKBKB
SCHEMBL15327834 0.74 CDC7 (0.46) IKBKBCHUKMAP2K1CLK4DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808086-B Heterocyclic substituted styryl-4-phenylpyridine derivative, preparation method and medical application thereof 上海海雁医药科技有限公司 2021-12-14 CN disclosed
CN-109956898-B Immunomodulator, preparation method and medical application thereof 上海海雁医药科技有限公司 2021-03-26 CN disclosed
CN-111808086-A Heterocyclic substituted styryl-4-phenylpyridine derivative, preparation method and medical application thereof 上海海雁医药科技有限公司 2020-10-23 CN disclosed
CN-109956898-A Immunomodulator and its preparation method and purposes pharmaceutically 上海海雁医药科技有限公司 2019-07-02 CN disclosed