SCHEMBL28308987

SCHEMBL28308987

CC(C)N1CCN(Cc2ccc3ccccc3n2)C(C)C1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.48
CYP1A2 P05177 1/20 0.40
HTR1A P08908 4/20 0.40
SLC6A4 P31645 3/20 0.40
DRD4 P21917 1/20 0.39
SLC6A9 P48067 1/20 0.39
PDE10A Q9Y233 1/20 0.39
HCRTR1 O43613 2/20 0.38
HCRTR2 O43614 2/20 0.38
FAAH O00519 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
ALOX5AP P20292 1/20 0.37
PDE2A O00408 1/20 0.37
CALCA P06881 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17460186 0.78 FAAH (0.52) CYP1A2HTR1ASLC6A4DRD4FAAH
SCHEMBL19281758 0.78 FAAH (0.52) CYP1A2HTR1ASLC6A4DRD4FAAH
SCHEMBL9963401 0.78 LMNA (0.45) HRH3CYP1A2DRD4SLC6A9
SCHEMBL9963404 0.78 LMNA (0.45) HRH3CYP1A2DRD4SLC6A9
SCHEMBL9963405 0.76 RAB9A (0.42) HRH3DRD4SLC6A9OPRK1
SCHEMBL19967980 0.76 SLC6A9 (0.49) HRH3SLC6A9
SCHEMBL17460429 0.74 CYP1A2 (0.43) CYP1A2HTR1ASLC6A4DRD4PDE10A
SCHEMBL17460275 0.74 CYP1A2 (0.43) CYP1A2HTR1ASLC6A4DRD4PDE10A
SCHEMBL3990929 0.69 FAAH (0.41) HRH3CYP1A2DRD4HCRTR1HCRTR2
SCHEMBL14197738 0.69 DRD4 (0.51) CYP1A2HTR1ADRD4PDE10AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814040-B The condensed 1,4- dihydro two of inhibitor as thermal excited transcryption factor 1 dislikes ene derivative 癌症研究科技有限公司 2019-07-30 CN disclosed