SCHEMBL283203

SCHEMBL283203

O=C(O)c1cc(Cl)ccc1F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.65
TP53 P04637 1/20 0.65
CA1 P00915 1/20 0.63
CA2 P00918 1/20 0.63
TSHR P16473 2/20 0.59
CASP1 P29466 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
MRGPRX4 Q96LA9 1/20 0.55
KDM4E B2RXH2 1/20 0.52
HSD17B10 Q99714 1/20 0.52
GRIK1 P39086 2/20 0.50
MYC P01106 2/20 0.50
NR4A1 P22736 1/20 0.50
F7 P08709 1/20 0.48
F3 P13726 1/20 0.48
KEAP1 Q14145 1/20 0.48
NFE2L2 Q16236 1/20 0.48
KMO O15229 2/20 0.47
ALB P02768 1/20 0.47
AKR1C4 P17516 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30396748 1.00 ALDH1A1 (0.65) ALDH1A1TP53CA1CA2TSHR
SCHEMBL392840 0.84 SMN1; SMN2 (0.63) ALDH1A1TP53CA1CA2TSHR
SCHEMBL28072667 0.84 ALDH1A1 (0.50) ALDH1A1TP53CA1CA2TSHR
SCHEMBL9692043 0.84 ALDH1A1 (0.50) ALDH1A1TP53CA1CA2TSHR
SCHEMBL30349584 0.82 ALDH1A1 (0.56) ALDH1A1TP53CA1CA2TSHR
SCHEMBL284068 0.82 ALDH1A1 (0.56) ALDH1A1TP53CA1CA2TSHR
SCHEMBL1000440 0.81 ALDH1A1 (0.71) ALDH1A1TP53CA1CA2TSHR
SCHEMBL19514758 0.81 ALDH1A1 (0.71) ALDH1A1TP53CA1CA2TSHR
SCHEMBL10965676 0.80 GRIK1 (0.54) ALDH1A1TP53CA1CA2TSHR
SCHEMBL3621421 0.80 MAOB (0.47) ALDH1A1TP53CA1CA2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 319 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114450275-B Heteroaryl aminopyridine alcohol derivatives and pharmaceutical composition for preventing or treating autoimmune diseases comprising the same as active ingredient 因诺沃治疗有限公司 2024-11-19 CN claimed
CN-113501807-A Tetrahydrobenzothiophene compound, and preparation method and application of pharmaceutical composition 重庆科技学院 2021-10-15 CN claimed
EP-3551633-B1 SUBSTITUTED PYRAZOLOAZEPIN-4-ONES AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS LEO PHARMA AS (DK) 2021-03-31 EP claimed
CN-111548325-A Preparation method of halogenated benzothiazepine compound, product prepared by preparation method and application of product 西安都创医药科技有限公司 2020-08-18 CN claimed
EP-3551633-A1 SUBSTITUTED PYRAZOLOAZEPIN-4-ONES AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS Leo Pharma A/S (DK) 2019-10-16 EP claimed
WO-2018108230-A1 SUBSTITUTED PYRAZOLOAZEPIN-4-ONES AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2018-06-21 WO claimed
EP-2379558-B1 NOVEL HETEROCYCLIC COMPOUNDS FOR USE AS METAP-2 INHIBITORS MERCK PATENT GMBH (DE) 2016-03-23 EP claimed
CN-104529735-A 1-(5-bromo-4-chloro-2-fluorophenyl)-ethanone synthesis method SUZHOU SHIYA BIOPHARMACEUTICALS INC 2015-04-22 CN claimed
US-20110281859-A1 NOVEL HETEROCYCLIC COMPOUNDS AS METAP-2 INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2011-11-17 US claimed
US-20110260051-A1 METHOD FOR DETECTING TRACER COMPOUNDS FOR HYDROCARBON PRODUCTION TOTAL S.A. (FR) 2011-10-27 US claimed
EP-3433239-B1 SMALL MOLECULE INHIBITORS OF THE NUCLEAR TRANSLOCATION OF ANDROGEN RECEPTOR FOR THE TREATMENT OF CASTRATION-RESISTANT PROSTATE CANCER UNIV PITTSBURGH COMMONWEALTH SYS HIGHER EDUCATION (US) 2026-05-27 EP disclosed
EP-3558298-B1 ANTIDIABETIC SPIROCHROMAN COMPOUNDS MERCK SHARP & DOHME LLC (US) 2026-03-11 EP disclosed
US-12338241-B2 Bicyclic sulfones and sulfoxides and methods of use thereof GENENTECH, INC. (US) 2025-06-24 US disclosed
CN-116655497-B Amidine derivative compound and preparation method and application thereof 中国科学院上海药物研究所 2025-06-03 CN disclosed
CN-114450275-B Heteroaryl aminopyridine alcohol derivatives and pharmaceutical composition for preventing or treating autoimmune diseases comprising the same as active ingredient 因诺沃治疗有限公司 2024-11-19 CN disclosed
WO-2003037346-A1 6-PHENYL-N-PHENYL-(1,3,5) -TRIAZINE-2,4-DIAMINE DERIVATIVES AND RELATED COMPOUNDS WITH LYSOPHPHOSPHATIDIC ACID ACYLTRANSFERASE BETA (LPAAT-BETA) INHIBITORY ACTIVITY FOR USE IN THE TREATMENT OF CANCER CELL THERAPEUTICS, INC. (US) 2003-05-08 WO disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed
EP-0295833-A1 Aromatic-Spiropiperidine oxazepinones (and thiones) A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1988-12-21 EP disclosed
US-4746655-A ANTIHISTAMINES A. H. ROBINS COMPANY, INCORPORATED (US) 1988-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12338241-B2 Bicyclic sulfones and sulfoxides and methods of use thereof RB1, CCNE2, RPS3A ALDH1A1 1912/4885TP53 64/4885CA1 2308/4885
US-20110281859-A1 NOVEL HETEROCYCLIC COMPOUNDS AS METAP-2 INHIBITORS METAP2, METAP1, XPNPEP2 ALDH1A1 1917/4885TP53 715/4885CA1 1303/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.