SCHEMBL2832259

SCHEMBL2832259

Cc1ccc(NC(=O)Oc2cnoc2C)cc1Nc1ncc(-c2ccncc2)o1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIT P10721 5/20 0.38
FLT1 P17948 5/20 0.38
FLT4 P35916 5/20 0.38
KDR P35968 5/20 0.38
ALOX5 P09917 1/20 0.36
IMPDH2 P12268 2/20 0.36
ABL1 P00519 3/20 0.35
PDGFRB P09619 2/20 0.35
BCR P11274 2/20 0.35
PDGFRA P16234 2/20 0.35
PRKCA P17252 1/20 0.34
P2RY1 P47900 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL544201 0.84 RAB9A (0.48) KITKDRIMPDH2ABL1PDGFRB
SCHEMBL543923 0.80 KIT (0.42) KITFLT1FLT4KDRALOX5
SCHEMBL13380736 0.78 KIT (0.43) KITFLT1FLT4KDRALOX5
SCHEMBL2831554 0.78 KIT (0.41) KITIMPDH2ABL1PDGFRBBCR
SCHEMBL5712004 0.77 SMN1; SMN2 (0.51) KITMEN1LMNAKMT2A
SCHEMBL544093 0.76 MEN1 (0.50) FLT1FLT4KDRABL1PDGFRB
SCHEMBL544627 0.76 ROCK2 (0.47) FLT1FLT4KDRMEN1LMNA
SCHEMBL543650 0.76 ALDH1A1 (0.42) KITFLT1FLT4KDRALOX5
SCHEMBL543758 0.75 PSEN1 (0.51) KITFLT1FLT4KDR
SCHEMBL5712010 0.75 MEN1 (0.54) FLT1FLT4KDRABL1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1684750-B1 2-AMINOARYLOXAZOLE COMPOUNDS AS TYROSINE KINASE INHIBITORS AB SCIENCE (FR) 2010-04-28 EP claimed