Piperazine

Piperazine

SCHEMBL28325908

C1CNCCN1.C=CNS(=O)(=O)C=C

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Piperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237667 0.84
Piperazine SCHEMBL28473412 0.69 LMNA (0.40)
SCHEMBL15337777 0.67 EPHX1 (0.39)
SCHEMBL29926690 0.67 KDM4E (0.33)
SCHEMBL10415474 0.66
Vinylsulfonic Acid SCHEMBL6281464 0.64 MEN1 (0.30)
SCHEMBL22042504 0.64
SCHEMBL3631213 0.63
SCHEMBL2040906 0.60 TGM2 (0.37)
SCHEMBL1291237 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110251680-B Piperazine divinyl sulfonamide linker and preparation method and application thereof 上海科技大学 2022-10-18 CN claimed
CN-110251680-A A kind of piperazines divinyl sulfonamides link and the preparation method and application thereof 上海科技大学 2019-09-20 CN claimed
CN-110251680-B Piperazine divinyl sulfonamide linker and preparation method and application thereof 上海科技大学 2022-10-18 CN disclosed
CN-110251680-B Piperazine divinyl sulfonamide linker and preparation method and application thereof 上海科技大学 2022-10-18 CN disclosed
CN-110251680-B Piperazine divinyl sulfonamide linker and preparation method and application thereof 上海科技大学 2022-10-18 CN disclosed
CN-110251680-A A kind of piperazines divinyl sulfonamides link and the preparation method and application thereof 上海科技大学 2019-09-20 CN disclosed
CN-110251680-A A kind of piperazines divinyl sulfonamides link and the preparation method and application thereof 上海科技大学 2019-09-20 CN disclosed
CN-110251680-A A kind of piperazines divinyl sulfonamides link and the preparation method and application thereof 上海科技大学 2019-09-20 CN disclosed