SCHEMBL28328504

SCHEMBL28328504

COc1ccc(C2CCN(CCF)CC2)cc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.47
KCNH2 Q12809 3/20 0.46
QDPR P09417 1/20 0.46
TLR9 Q9NR96 9/20 0.44
TLR7 Q9NYK1 8/20 0.44
TLR4 O00206 2/20 0.44
TLR3 O15455 2/20 0.44
TLR8 Q9NR97 2/20 0.44
CHEK1 O14757 1/20 0.44
CARM1 Q86X55 2/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL310239 0.90 QDPR (0.49) DRD2KCNH2QDPRTLR9TLR7
SCHEMBL520088 0.83 QDPR (0.64) KCNH2QDPRTLR9TLR7CHEK1
SCHEMBL28137144 0.82 QDPR (0.47) DRD2KCNH2QDPRTLR9TLR7
SCHEMBL28136364 0.81 KCNH2 (0.48) KCNH2QDPRTLR9TLR7TLR4
SCHEMBL310593 0.77 DRD2 (0.62) DRD2KCNH2QDPRSLC6A4
SCHEMBL519694 0.76 QDPR (0.52) DRD2KCNH2QDPRCHEK1SLC6A4
SCHEMBL2226718 0.76 CAMK2D (0.49) DRD2KCNH2QDPRTLR9TLR7
SCHEMBL18764021 0.76 EGFR (0.49) QDPRTLR9TLR7TLR4TLR3
SCHEMBL1285354 0.75 DRD2 (0.50) DRD2CARM1SLC6A4
SCHEMBL1264565 0.75 TUBB4A (0.53) QDPRTUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106536503-B A kind of tyrosine kinase inhibitor and application thereof 北京澳合药物研究院有限公司 2019-09-06 CN disclosed
CN-106536503-A Tyrosine kinase inhibitor and uses thereof 山东轩竹医药科技有限公司 2017-03-22 CN disclosed