SCHEMBL28328680

SCHEMBL28328680

O=C(O)Cc1c(-c2ccco2)nnn1Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
ADORA2A P29274 10/20 0.52
ADORA1 P30542 10/20 0.52
ADORA2B P29275 9/20 0.52
ADORA3 P0DMS8 7/20 0.52
TSHR P16473 3/20 0.49
HPGD P15428 2/20 0.45
IDO1 P14902 1/20 0.45
HSD17B10 Q99714 3/20 0.44
POLB P06746 1/20 0.44
RECQL P46063 1/20 0.44
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28343059 0.81 IDO1 (0.51) ALDH1A1TSHRHPGDIDO1POLB
SCHEMBL26817248 0.72 ALDH1A1 (0.56) ALDH1A1TSHRHPGDIDO1POLB
SCHEMBL28328763 0.71 CYP19A1 (0.48) ADORA2AADORA1ADORA2BADORA3HPGD
SCHEMBL28328678 0.71 PTGER4 (0.54) ALDH1A1ADORA3NPC1RAB9A
SCHEMBL28343588 0.70 KMT2A (0.50) ALDH1A1TSHRHPGDIDO1POLB
SCHEMBL28329962 0.70 PTGDR2 (0.41) HPGDIDO1POLBKDM4E
SCHEMBL28328682 0.70 TGM2 (0.44) ALDH1A1ADORA3KDM4E
SCHEMBL6357277 0.69 ALDH1A1 (1.00) ALDH1A1ADORA2AADORA1ADORA2BADORA3
SCHEMBL28878277 0.68 PTGDR2 (0.50) HPGDIDO1POLBRECQLKDM4E
SCHEMBL28329954 0.68 CNR2 (0.48) ALDH1A1POLBLMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110498773-B Method for synthesizing 1, 4-substituted 1,2, 3-triazole from acetylenic acid 乐山师范学院 2021-07-02 CN disclosed
CN-110526875-A A kind of acetylenic acid multicomponent synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-12-03 CN disclosed
CN-110498772-A A kind of Terminal Acetylenes multicomponent synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-11-26 CN disclosed
CN-110498773-A A kind of acetylenic acid synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-11-26 CN disclosed
CN-106866557-B (Z)-β-alkenyl bromine multicomponent prepares the method and application of 1,4- substitution -1,2,3- triazole 乐山师范学院 2019-11-12 CN disclosed