SCHEMBL28328752

SCHEMBL28328752

Clc1cc2ccccc2c(CBr)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.44
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.35
HIF1A Q16665 1/20 0.35
CYP1B1 Q16678 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HTR2A P28223 1/20 0.35
NQO2 P16083 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP2A6 P11509 2/20 0.34
CYP1A2 P05177 1/20 0.34
CCR1 P32246 1/20 0.34
CCR8 P51685 1/20 0.34
PTPN1 P18031 1/20 0.34
HTT P42858 2/20 0.34
USP2 O75604 1/20 0.34
MAPT P10636 1/20 0.34
ERBB2 P04626 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16516540 0.81 L3MBTL1 (0.44) L3MBTL1KMT2AALDH1A1HIF1ACYP1B1
SCHEMBL16008667 0.81 L3MBTL1 (0.44) L3MBTL1KMT2AALDH1A1HIF1ACYP1B1
SCHEMBL14693670 0.81 L3MBTL1 (0.44) L3MBTL1KMT2AALDH1A1HIF1ACYP1B1
SCHEMBL28327541 0.81 HTR2A (0.48) L3MBTL1KMT2AALDH1A1HIF1ACYP1B1
SCHEMBL9494876 0.80 ADORA3 (0.45) L3MBTL1ALDH1A1HIF1ACYP1B1HSD17B10
SCHEMBL31427619 0.78 ALDH1A1 (0.37) L3MBTL1KMT2AALDH1A1HIF1ACYP1B1
SCHEMBL10527114 0.77 L3MBTL1 (0.40) L3MBTL1KMT2AALDH1A1HIF1ACYP1B1
SCHEMBL27599861 0.77 L3MBTL1 (0.40) L3MBTL1KMT2AALDH1A1NQO2KDM4E
Bromide SCHEMBL5045247 0.76 ALDH1A1 (0.34) L3MBTL1ALDH1A1HIF1ACYP1B1HSD17B10
SCHEMBL28457078 0.75 MAPK1 (0.51) ALDH1A1KDM4ECYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113651820-A Urea compounds for dual IDO and TDO inhibitors 正大天晴药业集团股份有限公司 2021-11-16 CN disclosed
CN-110382500-B Urea compounds for dual IDO and TDO inhibitors 正大天晴药业集团股份有限公司 2021-08-10 CN disclosed
CN-110382500-A Carbamide compounds for IDO and TDO double inhibitor 正大天晴药业集团股份有限公司 2019-10-25 CN disclosed