SCHEMBL28342145

SCHEMBL28342145

Cc1c(N)cnc(N)c1[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
TP53 P04637 1/20 0.42
LMNA P02545 8/20 0.42
MAPT P10636 7/20 0.42
HTT P42858 5/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 2/20 0.41
MITF O75030 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PRMT1 Q99873 1/20 0.38
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3922708 0.85 PKM (0.42) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL10415524 0.85 ALDH1A1 (0.46) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL9131751 0.83 ALDH1A1 (0.41) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL31539746 0.81 MAPT (0.44) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL27961261 0.81 ALDH1A1 (0.38) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL203339 0.81 LMNA (0.43) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL2086204 0.81 MAPT (0.44) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL18937751 0.81 MAPT (0.36) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL202940 0.81 ALDH1A1 (0.40) ALDH1A1TP53LMNAMAPTHTT
SCHEMBL28191633 0.77 MAPT (0.44) ALDH1A1TP53LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117440945-A Pyrimidine or pyridine derivative, preparation method thereof and application thereof in pharmacy 上海和誉生物医药科技有限公司 2024-01-23 CN disclosed
CN-111892579-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-07-25 CN disclosed
CN-111875585-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-06-23 CN disclosed
CN-115867539-A 2, 3-dihydro-1H-pyrrolo [3,2-b ] pyridine derivatives, preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-28 CN disclosed
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
CN-110642838-B EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2022-08-09 CN disclosed
CN-110642836-B EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2022-08-09 CN disclosed
CN-111892579-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-06 CN disclosed
CN-111875585-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-03 CN disclosed
CN-106660993-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-09-11 CN disclosed
CN-110642836-A EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2020-01-03 CN disclosed
CN-110642838-A EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2020-01-03 CN disclosed