SCHEMBL28347669

SCHEMBL28347669

COC(=O)c1ccc2c[c]ccc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.40
CYP1A2 P05177 2/20 0.39
CNR2 P34972 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 3/20 0.38
HPGD P15428 1/20 0.38
KDM4E B2RXH2 2/20 0.38
HTT P42858 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPT P10636 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4850106 0.87 MAPK1 (0.40) MAPK1CYP1A2CNR2NPC1TP53
SCHEMBL6231133 0.81 MGAM (0.38) CNR2NPC1TP53RAB9ASMN1; SMN2
SCHEMBL3922658 0.78 PIM1 (0.41) CNR2RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL5873635 0.77 ALDH1A1 (0.61) NPC1TP53RAB9ASMN1; SMN2ALDH1A1
SCHEMBL530121 0.77 KMT2A (0.37) CYP1A2CNR2NPC1TP53RAB9A
SCHEMBL30208641 0.76 MGAM (0.61) CNR2RAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL725183 0.76 MGAM (0.61) CNR2RAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL16880740 0.75 HSD17B14 (0.51) CYP1A2NPC1TP53CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL30615167 0.75 MGAM (0.59) CNR2RAB9ASMN1; SMN2ALDH1A1HPGD
Hydrochloric Acid SCHEMBL16793838 0.75 MGAM (0.59) CNR2RAB9ASMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110563713-A 4-phenyl substituted isoxazole compound and application thereof in antihistamine medicine 王兴理 2019-12-13 CN claimed