SCHEMBL283482

SCHEMBL283482

NC(=NO)c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F7 P08709 1/20 0.59
F3 P13726 1/20 0.59
SARM1 Q6SZW1 1/20 0.59
SIRT2 Q8IXJ6 1/20 0.59
SIRT6 Q8N6T7 1/20 0.59
SIRT1 Q96EB6 1/20 0.59
SIRT3 Q9NTG7 1/20 0.59
SIRT5 Q9NXA8 1/20 0.59
SIRT4 Q9Y6E7 1/20 0.59
POLB P06746 2/20 0.52
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
APP P05067 1/20 0.50
GAA P10253 1/20 0.50
HCAR3 P49019 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
HTT P42858 1/20 0.49
NPC1 O15118 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312479 1.00 F7 (0.59) F7F3SARM1SIRT2SIRT6
SCHEMBL29692126 1.00 F7 (0.59) F7F3SARM1SIRT2SIRT6
SCHEMBL283480 1.00 F7 (0.59) F7F3SARM1SIRT2SIRT6
Hydrochloric Acid SCHEMBL28676955 0.98 F7 (0.57) F7F3SARM1SIRT2SIRT6
Niacin SCHEMBL9231503 0.89 ALDH1A1 (0.70) F7F3SARM1SIRT2SIRT6
SCHEMBL834568 0.83 F7 (0.59) F7F3SARM1SIRT2SIRT6
SCHEMBL27764447 0.83 F7 (0.59) F7F3SARM1SIRT2SIRT6
SCHEMBL24170739 0.82 F7 (0.57) F7F3SARM1SIRT2SIRT6
SCHEMBL5056593 0.79 CYP3A4 (0.54) F7F3SARM1SIRT2SIRT6
SCHEMBL22281477 0.79 CYP3A4 (0.54) F7F3SARM1SIRT2SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 211 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3978219-A NICOTINAMIDOXIME AS AN ANTI-INFLAMMATORY AGENT STAUFFER CHEMICAL COMPANY (US) 1976-08-31 US claimed
US-20260042731-A1 (2,4-DICHLOROPHENOXY)ACETIC ACID ANALOGS CORTEVA AGRISCIENCE LLC (US) 2026-02-12 US disclosed
EP-4363415-B1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS TECNIMEDE SOCIEDADE TECNICO MEDICINAL SA (PT) 2025-12-10 EP disclosed
US-12478621-B2 Substituted aminoquinolones as dgkalpha inhibitors for immune activation DEUTSCHES KREBSFORSCHUNGSZENTRUM (DE) 2025-11-25 US disclosed
EP-3885340-B1 ANDROGEN RECEPTOR MODULATING COMPOUNDS ORION CORP (FI) 2024-11-27 EP disclosed
US-20240279217-A1 Heterocyclic compounds for the treatment of tuberculosis TECNIMEDE - Sociedade Técnico-medicinal, SA (PT) 2024-08-22 US disclosed
US-11998539-B2 Substituted aminoquinolones as DGKalpha inhibitors for immune activation BAYER AKTIENGESELLSCHAFT (DE) 2024-06-04 US disclosed
EP-4363415-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS Tecnimede, Sociedade Técnico-Medicinal, SA (PT) 2024-05-08 EP disclosed
CN-117813004-A Auxin herbicide and application method thereof 科迪华农业科技有限责任公司 2024-04-02 CN disclosed
WO-2024031002-A1 (2,4-DICHLOROPHENOXY)ACETIC ACID ANALOGS CORTEVA AGRISCIENCE LLC (US) 2024-02-08 WO disclosed
EP-0604352-A2 Aryl substituted heterocyclic compounds NEUROSEARCH A/S (DK) 1994-06-29 EP disclosed
US-5317103-A Migraine treatment MERCK SHARP & DOHME LIMITED (GB) 1994-05-31 US disclosed
EP-0438230-A2 Indole-substituted five-membered heteroaromatic compounds MERCK SHARP & DOHME LTD. (GB) 1991-07-24 EP disclosed
US-4308399-A O-(3-Amino-2-hydroxy-propyl)-amidoxime derivatives, process for the preparation thereof and pharmaceutical compositions containing same CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1981-12-29 US disclosed
US-4305948-A N-Hydroxy-1,2-dihydro-2-oxo-5-(pyridinyl)-nicotinimidamide and their cardiotonic use STERLING DRUG INC. (US) 1981-12-15 US disclosed
US-4187220-A New O-(3-amino-2-hydroxy-propyl)-amidoxime derivatives, process for the preparation thereof and pharmaceutical compositions containing same CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA R.T. (HU) 1980-02-05 US disclosed
US-4065563-A 3-Hetero-5-isothiocyanophenyl oxadiazoles as antifungal and antibacterial agents E. R. SQUIBB & SONS, INC. (US) 1977-12-27 US disclosed
US-4022901-A FUNGICIDAL AND BACTERICIDAL ACTIVITY E. R. SQUIBB & SONS, INC. (US) 1977-05-10 US disclosed
US-3978219-A NICOTINAMIDOXIME AS AN ANTI-INFLAMMATORY AGENT STAUFFER CHEMICAL COMPANY (US) 1976-08-31 US disclosed
US-3978219-A NICOTINAMIDOXIME AS AN ANTI-INFLAMMATORY AGENT STAUFFER CHEMICAL COMPANY (US) 1976-08-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240279217-A1 Heterocyclic compounds for the treatment of tuberculosis SDHA, NQO1, FNTB F7 4412/4885F3 4496/4885SARM1 1194/4885
US-12478621-B2 Substituted aminoquinolones as dgkalpha inhibitors for immune activation DGKK, DGKG, DGKA F7 2632/4885F3 587/4885SARM1 1574/4885
US-11998539-B2 Substituted aminoquinolones as DGKalpha inhibitors for immune activation DGKK, DGKG, DGKA F7 2632/4885F3 587/4885SARM1 1574/4885
US-20260042731-A1 (2,4-DICHLOROPHENOXY)ACETIC ACID ANALOGS DDT, AADAC, HACL2 F7 2245/4885F3 4081/4885SARM1 1282/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.