SCHEMBL28348308

SCHEMBL28348308

O=C(NCCc1ccncc1)c1csc(-c2cccnc2)n1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.65
HPGD P15428 2/20 0.61
TSHR P16473 1/20 0.61
HDAC2 Q92769 1/20 0.60
TP53 P04637 1/20 0.60
MAPT P10636 1/20 0.60
IRAK4 Q9NWZ3 3/20 0.60
ALDH1A1 P00352 4/20 0.59
KDM4E B2RXH2 2/20 0.59
TLR7 Q9NYK1 1/20 0.58
RAB9A P51151 3/20 0.57
ATM Q13315 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
POLB P06746 1/20 0.57
ALOX15 P16050 1/20 0.57
HTT P42858 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
NPC1 O15118 2/20 0.56
LMNA P02545 1/20 0.56
THRB P10828 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703958 0.93 IRAK4 (0.66) HDAC6HPGDTSHRHDAC2TP53
SCHEMBL28348018 0.91 HPGD (0.63) HDAC6HPGDHDAC2MAPTALDH1A1
SCHEMBL28601973 0.85 HDAC6 (0.69) HDAC6HPGDTSHRHDAC2TP53
SCHEMBL28344825 0.84 IRAK4 (0.68) HDAC6HPGDTSHRHDAC2TP53
SCHEMBL17175809 0.81 IRAK4 (0.69) HDAC6HPGDHDAC2TP53MAPT
SCHEMBL28970478 0.80 HDAC6 (0.78) HDAC6HDAC2MAPTIRAK4ALDH1A1
SCHEMBL11114421 0.80 HPGD (0.67) HDAC6HPGDMAPTTLR7RAB9A
SCHEMBL3477450 0.79 HDAC6 (0.67) HDAC6HDAC2MAPTIRAK4TLR7
SCHEMBL2113234 0.79 HDAC6 (0.67) HDAC6HDAC2TP53MAPTIRAK4
SCHEMBL24755152 0.79 HDAC6 (1.00) HDAC6HDAC2MAPTIRAK4TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110407824-B Aryl formamide compound and preparation method, pharmaceutical composition and application thereof 安徽医科大学 2021-07-02 CN disclosed
CN-110407824-A Aryl methanamide compounds and preparation method thereof, pharmaceutical composition and purposes UNIV ANHUI MEDICAL 2019-11-05 CN disclosed