SCHEMBL7703958

SCHEMBL7703958

O=C(NCCc1ccccc1)c1csc(-c2cccnc2)n1

nearest known ligand 0.89

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 3/20 0.66
MAPT P10636 2/20 0.66
TP53 P04637 1/20 0.66
HDAC6 Q9UBN7 1/20 0.65
TLR7 Q9NYK1 1/20 0.61
ALDH1A1 P00352 4/20 0.61
KDM4E B2RXH2 2/20 0.61
HDAC2 Q92769 1/20 0.60
HIF1A Q16665 1/20 0.60
RAB9A P51151 3/20 0.59
NPC1 O15118 2/20 0.59
GAA P10253 1/20 0.59
LMNA P02545 1/20 0.59
HPGD P15428 2/20 0.58
TSHR P16473 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
ATM Q13315 1/20 0.57
POLB P06746 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28348308 0.93 HDAC6 (0.65) IRAK4MAPTTP53HDAC6TLR7
SCHEMBL17175809 0.88 IRAK4 (0.69) IRAK4MAPTTP53HDAC6TLR7
SCHEMBL28344825 0.86 IRAK4 (0.68) IRAK4MAPTTP53HDAC6TLR7
SCHEMBL28601973 0.85 HDAC6 (0.69) IRAK4MAPTTP53HDAC6TLR7
SCHEMBL28348018 0.83 HPGD (0.63) MAPTHDAC6ALDH1A1HDAC2HIF1A
SCHEMBL11910582 0.82 MAPT (0.64) MAPTTP53HDAC6TLR7ALDH1A1
SCHEMBL28970478 0.80 HDAC6 (0.78) IRAK4MAPTHDAC6TLR7ALDH1A1
Chlorobenzene SCHEMBL28344826 0.80 HDAC2 (0.67) IRAK4MAPTTP53HDAC6TLR7
SCHEMBL2113234 0.79 HDAC6 (0.67) IRAK4MAPTTP53HDAC6TLR7
SCHEMBL3477450 0.79 HDAC6 (0.67) IRAK4MAPTHDAC6TLR7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed