SCHEMBL28348347

SCHEMBL28348347

C#CSc1ccc(F)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
ACHE P22303 1/20 0.35
PYCR1 P32322 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
PTGS1 P23219 1/20 0.33
FBP1 P09467 1/20 0.32
IDO1 P14902 1/20 0.31
ORAI1 Q96D31 1/20 0.31
ORAI2 Q96SN7 1/20 0.31
ORAI3 Q9BRQ5 1/20 0.31
TRPV6 Q9H1D0 1/20 0.31
CYP1A2 P05177 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CES2 O00748 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL469852 0.76 ALDH1A1 (0.52) MAOAMAOBCA1CA2CA7
SCHEMBL7557350 0.72 LMNA (0.44) MAOAMAOBPYCR1ALDH1A1IDO1
SCHEMBL315215 0.71
SCHEMBL576260 0.69 MEN1 (0.48) CA1CA2CA7CA9ACHE
SCHEMBL223757 0.69 FBP1 (0.52) MAOAMAOBCA1CA2CA7
Ethyne SCHEMBL27932680 0.67 CA1 (0.53) CA1CA2CA7CA9ACHE
SCHEMBL15199481 0.67
SCHEMBL6597844 0.67
SCHEMBL13499 0.67
SCHEMBL7567051 0.65 ACACB (0.45) MAOAMAOBALDH1A1MAPK1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110724110-B Preparation method and application of 4-heteroatom-3, 4,5 substituted isoxazole compound 香港科技大学深圳研究院 2022-04-26 CN disclosed
CN-110724110-A Preparation method and application of 3,4,5 (4-heteroatom) fully-substituted isoxazole compound 香港科技大学深圳研究院 2020-01-24 CN disclosed