SCHEMBL28355273

SCHEMBL28355273

Cc1c(N)c(N)nc(OCC(F)(F)F)c1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.37
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
USP2 O75604 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
THRB P10828 1/20 0.35
G6PD P11413 1/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MBOAT4 Q96T53 3/20 0.34
MAPK1 P28482 1/20 0.34
NUDT1 P36639 2/20 0.33
SCN9A Q15858 1/20 0.33
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704969 0.71 HSP90AA1 (0.47) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL13575846 0.70 PIK3CA (0.41) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL10569355 0.67 ALDH1A1 (0.45) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL2947663 0.67 ALDH1A1 (0.46) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL21756757 0.67 ALDH1A1 (0.42) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL18072509 0.67 NUDT1 (0.73) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL30819099 0.66 MAPT (0.37) ALDH1A1MAPTKMT2AL3MBTL1CNR2
SCHEMBL11581915 0.66 LMNA (0.39) ALDH1A1KDM4E
SCHEMBL16097791 0.66 MEN1 (0.39) ADORA2AALDH1A1MAPTMEN1KMT2A
SCHEMBL13745731 0.66 ADORA2A (0.40) ADORA2AALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110642838-B EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2022-08-09 CN disclosed
CN-110642838-A EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2020-01-03 CN disclosed