SCHEMBL28356802

SCHEMBL28356802

Cc1ccccc1-c1ccc(C=O)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.49
BACE1 P56817 1/20 0.49
LCK P06239 1/20 0.47
KDR P35968 1/20 0.47
JAK3 P52333 1/20 0.47
MAPK14 Q16539 1/20 0.47
TSHR P16473 8/20 0.46
ALDH1A1 P00352 7/20 0.46
CLK4 Q9HAZ1 8/20 0.44
CYP1A2 P05177 7/20 0.44
CYP3A4 P08684 7/20 0.44
CYP2C19 P33261 7/20 0.44
CYP2D6 P10635 5/20 0.44
MAPK1 P28482 3/20 0.44
CYP2C9 P11712 2/20 0.44
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MCL1 Q07820 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3689077 0.80 ALOX5AP (0.46) CTSDBACE1LCKKDRJAK3
SCHEMBL5737521 0.80 MCL1 (0.54) CTSDBACE1LCKKDRJAK3
SCHEMBL12999319 0.78 ALDH1A1 (0.50) CTSDBACE1LCKKDRJAK3
SCHEMBL5735316 0.78 ALDH1A1 (0.51) TSHRALDH1A1NPC1RAB9A
SCHEMBL14475320 0.77 CRHBP (0.45) BACE1ALDH1A1MAPK1LMNANPC1
SCHEMBL3971606 0.77 MCL1 (0.58) TSHRALDH1A1MCL1
SCHEMBL1767888 0.76 CYP1A2 (0.57) CTSDBACE1LCKKDRJAK3
SCHEMBL7936530 0.74 ERN1 (0.51) TSHRALDH1A1MEN1KMT2A
SCHEMBL5157768 0.73 CTSD (0.60) CTSDBACE1LCKKDRJAK3
SCHEMBL5711185 0.72 TSHR (0.58) TSHRALDH1A1CYP1A2CYP2C19CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110799509-A PD-1/PD-L1 inhibitors 吉利德科学公司 2020-02-14 CN disclosed