SCHEMBL28358263

SCHEMBL28358263

O=C(NOc1cccc(-c2ccccc2)c1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.53
HDAC2 Q92769 3/20 0.52
POLB P06746 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
HDAC1 Q13547 2/20 0.49
MRGPRX4 Q96LA9 1/20 0.49
HDAC3 O15379 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
KMO O15229 1/20 0.49
CTDSP1 Q9GZU7 1/20 0.49
BCL2L1 Q07817 1/20 0.48
MCL1 Q07820 1/20 0.48
TRPV1 Q8NER1 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
SMPD1 P17405 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL126697 0.84 ALDH1A1 (0.59) HDAC8HDAC2POLBKMT2AMEN1
SCHEMBL20299899 0.78 RXRA (0.49) HDAC2HDAC1MRGPRX4NPC1RAB9A
SCHEMBL6557528 0.75 NPC1 (0.55) HDAC8POLBKMT2AHDAC1MRGPRX4
SCHEMBL6555987 0.75 NPSR1 (0.51) HDAC8HDAC2POLBKMT2AMEN1
SCHEMBL17336876 0.75 HDAC8 (0.64) HDAC8POLBKMT2AMEN1NPC1
SCHEMBL7175937 0.74 ALOX5 (0.66) KMT2AMEN1MRGPRX4KMOALDH1A1
SCHEMBL29251267 0.74 KMT2A (0.52) HDAC8HDAC2POLBKMT2AMEN1
SCHEMBL27800573 0.72 NPC1 (0.56) HDAC2POLBKMT2AMEN1HDAC1
SCHEMBL27634795 0.72 JAK2 (0.56) HDAC2POLBKMT2AMEN1NPC1
SCHEMBL15901856 0.72 KAT6A (0.61) HDAC8HDAC1HDAC3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110818598-A Cathepsin inhibitor and preparation method and application thereof 沈阳药科大学 2020-02-21 CN disclosed