SCHEMBL2835871

SCHEMBL2835871

O=C1CCNCc2sccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 2/20 0.52
HRH1 P35367 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
CES1 P23141 1/20 0.34
MAP2K1 Q02750 2/20 0.34
APEX1 P27695 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
CASP1 P29466 1/20 0.33
MPI P34949 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1747122 0.74
SCHEMBL23426452 0.71 USP2 (0.52) CES1MAP2K1MEN1KMT2AALDH1A1
SCHEMBL3147129 0.71 USP2 (0.52) CES1MAP2K1MEN1KMT2AALDH1A1
SCHEMBL153954 0.71 USP2 (0.47) CES1MAP2K1MEN1KMT2AALDH1A1
SCHEMBL11088 0.71
Iodide SCHEMBL30536887 0.69 PNMT (0.69) PNMTCD44MAOB
Hydrochloric Acid SCHEMBL1427992 0.69 PNMT (0.69) PNMTCD44MAOB
SCHEMBL13441 0.69
SCHEMBL8171311 0.67
Bromide SCHEMBL28557676 0.67 PNMT (0.95) PNMTCD44MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US disclosed
US-20100048537-A1 HETEROARYL DERIVATIVES NIPPON SHINYAKU CO., LTD. (JP) 2010-02-25 US disclosed
EP-2141168-A1 HETEROARYL DERIVATIVES Nippon Shinyaku Co., Ltd. (JP) 2010-01-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048537-A1 HETEROARYL DERIVATIVES OPRD1, OPRM1, OPRK1 PNMT 1313/4885HRH1 550/4885HRH4 533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.