SCHEMBL28359192

SCHEMBL28359192

Cc1cc2cc(-c3ccccc3)cc(N)c2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
NPY5R Q15761 1/20 0.39
MAPT P10636 4/20 0.39
CASP1 P29466 2/20 0.39
AURKA O14965 1/20 0.39
THRB P10828 1/20 0.39
TTK P33981 1/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 4/20 0.38
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28359047 0.82 AURKA (0.47) NPY5RMAPTAURKATTKAURKB
SCHEMBL29635205 0.82 AURKA (0.47) NPY5RMAPTAURKATTKAURKB
SCHEMBL28358921 0.73 CRHBP (0.51) MAPTALDH1A1HSD17B10XDHNPC1
SCHEMBL6194760 0.72 PARP1 (0.46) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL3006008 0.71 NPY5R (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10492510 0.71 MAPT (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL31078313 0.71 HRH4 (0.46) ALDH1A1HPGDGAAHTTLMNA
SCHEMBL28796378 0.71 CYP2A6 (0.37) HPGDLMNACYP2A6KEAP1
SCHEMBL5797966 0.69 PTGS2 (0.60) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL6960951 0.68 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110818609-A Preparation method and application of 3-acetyl indole BRPF1 inhibitor 中国药科大学 2020-02-21 CN disclosed