SCHEMBL28360665

SCHEMBL28360665

C=CCN(C(C)=O)c1ccc(C#N)cc1I

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.36
ALB P02768 1/20 0.36
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
PGR P06401 1/20 0.32
SETDB1 Q15047 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
MAP2K1 Q02750 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
NSD2 O96028 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28360723 0.81 KDM4E (0.36) KDM4EALDH1A1
SCHEMBL28357008 0.80 FSCN1 (0.42) ALDH1A1MAPT
SCHEMBL28360698 0.76 TSHR (0.40) KDM4EALDH1A1
SCHEMBL28360711 0.75 HTT (0.44) KDM4EALDH1A1MAPT
SCHEMBL28360720 0.72 KDM4E (0.36) KDM4EALDH1A1
SCHEMBL28883288 0.71 SMN1; SMN2 (0.39) TTR
SCHEMBL28356849 0.71 ALDH1A1 (0.40) ALDH1A1MAPT
SCHEMBL4300629 0.68 TTR (0.47) TTRALBPGRKDM4EALDH1A1
SCHEMBL13283750 0.67 MAP2K1 (0.51) TTRALBMAP2K1
SCHEMBL2521954 0.67 TTR (0.40) TTRALBMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110804008-A 1, 3-disubstituted indoline derivative and preparation method thereof 陕西科技大学 2020-02-18 CN disclosed